Leveraging macrocyclic peptides to achieve novel MOAs and high specificity against intracellular targets

Time: 2:30 pm
day: Conference Day 2


  • Extensive scaffold hopping and physicochemical property tuning of display technology hits.
  • Generation of compounds with low and sub pM affinities and potent cell activity. 
  • Exploration of Unnatural Product’s parallel synthesis and computational design platform